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Gastrointestinal Pharmacology Study Guide

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Gastrointestinal Pharmacology Study Guide
Indication
Class/Target
Drugs
MOA
Appetite Stimulants
Anti Serotonin
Ghrelin agonist
Benzodiazepines
Cannabinoid
Anabolic steroids
Glucocorticoids
Vitamin Bs
Mirtazapine, Cyproheptadine
Capromorelin
Oxazepam
Dronabinol
Boldenone, Stanazolol
Pred, Dex, etc
B Vitamins
Inhibit serotonin receptor (5-HT2 for appetite)
Ghrelin agonist
GABA agonist
CB agonist
Stim orexigenic center?
?
?
Emetics
Central
Peripheral
Apomorphine (dogs!)
Xylazine (cats!)
Sodium chloride
Syrup of Ipecac
Hydrogen peroxide
Dop agonist CRTZ
α-2 agonist
reflex vomit
GI irritant
GI irritant
Antiemetics
Antidopamine
Antihistamine
Antiserotonin
Antisubstance P
Phenothiazines
Metoclopramide (also prokinetic)
Dimenhydrinate, Diphenhydramine,
Meclizine (Motion sickness only)
Ondansetron, Mirtazapine
Maropitant (So popular!)
Block D2 rec CRTZ
Block D2 rec, 5HT3 at high doses
Block H1,M1(vestibular)
Block 5HT3
Block NK1 rec
Anti-ulcer
Proton pump inhibit
H2 antagonists
Cytoprotectants
Omeprazole (PO), pantoprazole (IV)
Famotidine>rantidine>cimetidine
Misoprostol
Sucralfate
H+/K+ATPase inhibit
Inhibits H2 receptor
PGE analog
Polymerizes w/ ulcer
Prokinetics
Macrolide antibiotic
D2 antagonist
D2 antagonist
5HT4 rec agonist
Local anesthetic
Cholinergic stimulants
Cholinergic stimulant
Erythromycin
Metoclopramide
Domperidone
Cisapride
Lidocaine
Bethanecol, pilocarpine
Neostigmine
Motilin rec agonist
D2-, 5HT4+
D2-
5HT4+
? equine ileus use
Direct parasympathomimetics
Indirect parasympathomimetic
Laxatives
Bulk (fiber supplem)
Hyperosmotic
Methylcellulose, psyllium, bran, pumpkin
Lactulose, magn hydroxide
Psyllium: equine sand colic
Draw water into bowel
Anti-diarrheals
(acute diarrhea)
Opioids (use is questionable)
Anticholinergic
loperamide, paregoric, diphenyloxylate,
N-butylscopolamine
Decrease propulsive motility
blunt prop& segmental motility;
antispasmodic for equine gas colic

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Gastrointestinal Pharmacology – Study Guide Indication Class/Target Appetite Stimulants Anti Serotonin Ghrelin agonist Benzodiazepines Cannabinoid Anabolic steroids Glucocorticoids Vitamin Bs Emetics Central Peripheral Antiemetics Antidopamine Antihistamine Anti-ulcer Prokinetics Laxatives Anti-diarrheals (acute diarrhea) Antiserotonin Antisubstance P Proton pump inhibit H2 antagonists Cytoprotectants Macrolide antibiotic D2 antagonist D2 antagonist 5HT4 rec agonist Local anesthetic Cholinergic stimulants Cholinergic stimulant Bulk (fiber supplem) Hyperosmotic Opioids (use is questiona ...
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